Available GPCR and other cell lines
U-PHARM
Laboratories LLC
Accelerate drug discovery
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1001 Adenosine A2a Receptor
1002 Adenosine A2b Receptor
1003 Adenylate Cyclase Activating Polypeptide 1Receptor (ADCYAP1R1)
1004 Amylin 3 Receptor
1005 Arginine Vasopressin 2 Receptor (AVPR2)
1006 Beta-1 Adrenergic Receptor (ADRB1)
1007 Beta-2 Adrenergic Receptor (ADRB2)
1008 Calcitonin Receptor (CALCR)
1009 Calcitonin-like Receptor (CALCRL)
1010 Corticotropin Releasing Hormone Receptor 1 (CRHR1)
1011 Corticotropin Releasing Hormone Receptor 2 (CRHR2)
1012 Dopamine Receptor 1 (DRD1)
1013 Dopamine Receptor 5 (DRD5)
1014 Follicle Stimulating Hormone Receptor (FSHR)
1015 Gastric Inhibitor Peptide Receptor(GIPR)
1016 Glucagon Receptor (GCGR)
1017 Glucagon-like Receptor 1 (GLP1R)
1018 Glucagon-like Receptor 2 (GLP2R)
1019 Melanocortin 1 Receptor (MC1R)
1020 Melanocortin 3 Receptor (MC3R)
1021 Melanocortin 4 Receptor (MC4R)
1022 Melanocortin 5 Receptor (MC5R)
1023 Parathyroid Hormone Receptor 1 (PTHR1)
1024 Parathyroid Hormone Receptor 2 (PTHR2)
1025 Prostaglandin D Receptor 2 (PTGDR2)
1026 PTGER2 (EP2)
1027 Prostaglandin E Receptor 4 (PTGER4)
1028 Prostaglandin I2 Receptor (PTGIR)
1029 Secretin Receptor (SCTR)
1030 Serotonin Receptor 4 (HTR4)
1031 Serotonin Receptor 6 (HTR6)
1032 Serotonin Receptor Receptor 7 (HTR7)
1033 Thyroid Stimulating Hormone Receptor (TSHR)
1034 Vasoactive Intestinal Peptide Receptor 1 (VIPR1)
1035 Vasoactive Intestinal Peptide Receptor 2 (VIPR2)
Gi-coupled receptors with cyclic nucleotide-gated (CNG) channels
1036 Adenosine A1 Receptor
1037 Adenosine A3 Receptor
1038 Angiotensin Receptor-like 1
1039 Cannabinoid Receptor 1
1040 Cannabinoid Receptor 2
1041 Chemokine (C-C motif) Receptor 5
1042 Chemokine (C-X-C motif) Receptor 4
1043 Dopamine Receptor 2 (DRD2)
1044 Glutamate Receptor, Metabotropic 2
1045 Glutamate Receptor, Metabotropic 4
1046 Glutamate Receptor, Metabotropic 7
1047 Glutamate Receptor, Metabotropic 8
1048 Melanin Concentrating Hormone Receptor 1 (MCHR1)
1049 Neuropeptide Y Receptor Y1 (NPY1R)
1050 Neuropeptide Y Receptor Y2 (NPY2R)
1051 Neuropeptide Y Receptor Y4 (NPY4R)
1052 Opiate Receptor-like 1 (ORL1)
1053 Opioid receptor, kappa 1
1054 Opioid receptor, Mu
1055 Somatostatin Receptor 5 (SSTR5)
1056 Sphingolipid G-protein-coupled receptor 1 (EDG1)
Transduced PDEs with cyclic nucleotide-gated (CNG) channels
1057 Phosphodiesterase 4
1058 Phosphodiesterase 2A, cGMP-stimulated, (PDE2A)
Gq-coupled receptors
1059 Histamine receptor 1 (H1)
1060 Alpha adrenergic receptor 1B
Promiscuous and chimeric G proteins, with or without GPCRs
1061 G16
1062 Gqi1
1063 Gqi3
1064 Gqz
1065 Gsi1
1066 Melanin Concentrating Hormone Receptor 1 (MCHR1) + Gqi3
1067 Adenosine A3 Receptor + Gqi1
Reporter genes
1068 Luciferase reporter gene
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